All::Respiratory::Pharmacology::H1-receptor antagonists

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What is the method of action of H1-receptor antagonists?

H1 receptors, histamine induces the features of immediate-type (type 1) hypersensitivity

H1-receptor antagonists

What is the main clinical use of H1-receptor antagonists?

  • Allergies, particularly hay fever
  • To aid relief of pruritus and urticaria
  • Adjunctive treatment in anaphylaxis

H1-receptor antagonists

What are the main contraindications of H1-receptor antagonists?

severe liver disease

H1-receptor antagonists

Why do first-generation H1-receptor antagonists cause sedation?

They cross the blood brain barrier and H1 receptors, has a role in the brain in maintaining wakefulness

H1-receptor antagonists

What is an example of a first-generation H1-receptor antagonists?

chlorphenamine

H1-receptor antagonists

What is an example of a second-generation H1-receptor antagonists?

loratadine, cetirizine and fexofenadine

H1-receptor antagonists